Dr. Mohammad  Emad Azab

Dr. Mohammad Emad Azab

Professor
Ain Shams University, Egypt


Highest Degree
Ph.D. in Organic Chemistry from Ain Shams University, Cairo, Egypt

Share this Profile

Area of Interest:

Chemistry
100%
Organic Chemistry
62%
Chemical Biology
90%
Analysis of Chemicals
75%
Active Compounds
55%

Selected Publications

  1. Anwer, K.E., G.H. Sayed, H.H. Hassan and M.E. Azab, 2019. Conventional and microwave synthesis of some new pyridine derivatives and evaluation their antimicrobial and cytotoxic activities. Egypt. J. Chem., Vol. 62. 10.21608/EJCHEM.2018.5115.1452.
    CrossRef  |  Direct Link  |  
  2. Sayed, G.H., M.E. Azab, N.A. Negm and K.E. Anwer, 2018. Antimicrobial and cytotoxic activities of some novel heterocycles bearing pyrazole moiety. J. Heterocyclic Chem., 55: 1615-1625.
    CrossRef  |  Direct Link  |  
  3. Sayed, G.H., M.E. Azab, K.E. Anwer, M.A. Raouf and N.A. Negm, 2018. Pyrazole, pyrazolone and enaminonitrile pyrazole derivatives: Synthesis, characterization and potential in corrosion inhibition and antimicrobial applications. J. Mol. Liquids, 252: 329-338.
    CrossRef  |  Direct Link  |  
  4. Fayed, A.A., S.A. Bahshwan, R.E. Abde-Megeid, M.E. Azab, A.E.G.E. Amr and M.M. Abdalla, 2018. Follicle-stimulating hormone (FSH) activities of some synthesized isoxazole and pyrazoline derivatives. Biomed. Res., 29: 3483-3491.
    Direct Link  |  
  5. Azab, M.E., S.S. Abdel‐Wahab, N.F. Mahmoud and G.A. Elsayed, 2018. Novel bridgehead thiadiazolopyrimidine derivatives with antimicrobial and antitumor activities. J. Heterocyclic Chem., 55: 2349-2359.
    CrossRef  |  Direct Link  |  
  6. Al Thagfan, S.S., A.A. Fayed, S.A. Bahshwan, A.E.G.E. Amr and N. Aljuhani et al., 2018. Pharmacological activities of some synthesized chiral macrocyclic pentapeptide Schiff base candidates. Biomed. Res., 29: 3605-3609.
    Direct Link  |  
  7. Madkour, H.F., M.E. Azab, A.F. Aly and M.S.M. Khamees, 2017. Novel heterocycles based on 1,3,4-thiadiazole scaffold as insecticides. J. Environ. Sci., 40: 19-44.
  8. Sayed, G.H., N.A. Negm, M.E. Azab and K.E. Anwer, 2016. Synthesis, characterization and biological activity of some pyrazole-pyrazolone derivatives. Egypt. J. Chem., 59: 663-672.
  9. Sayed, G.H., M.E. Azab, N.A. Negm and K.E. Anwer, 2016. Utility of enaminonitrile in the synthesis of novel heterocycles bearing pyrazole moiety and their antimicrobial and cytotoxic activity assessment. Al-Azhar Univ. Bull. Sci., 27: 9-22.
    CrossRef  |  Direct Link  |  
  10. El‐Hashash, M.A., M.E. Azab and J.M. Morsy, 2016. One‐pot synthesis of some dynamic 2‐substituted benzoxazinones and their corresponding qinazolinones of anticipated biological activity. J. Heterocyclic Chem., 53: 95-101.
    CrossRef  |  Direct Link  |  
  11. El-Hashash, M.A., M.E. Azab, R.A. Faty and A.E.E. Amr, 2016. Synthesis, antimicrobial and anti-inflammatory activity of some new benzoxazinone and quinazolinone candidates. Chem. Pharm. Bull., 64: 263-271.
    CrossRef  |  Direct Link  |  
  12. El-Hashash, M., J.M. Morsy, M.E. Azab and N. Mahmoud, 2016. Design, synthesis and anticancer activity of novel 2,3-and 2,4-disubstituted quinazoline and quinazolinone derivatives. Heterocycles, 92: 316-329.
  13. Azab, M.E., S.A. Rizk and N.F. Mahmoud, 2016. Facile synthesis, characterization and antimicrobial evaluation of novel heterocycles, schiff bases and N-nucleosides bearing phthalazine moiety. Chem. Pharm. Bull., 64: 439-450.
    CrossRef  |  Direct Link  |  
  14. Azab, M.E., N.M. Khalifa, A.A. Sediek, N.M. Sabry, M.M. Al-Omar and A.E.E. Amr, 2016. Synthesis and characterization of some new N-glycosides of pyridine-2,6-bis-carboxamides derivatives. Nucleosides Nucleotides Nucleic Acids, 35: 435-444.
    CrossRef  |  Direct Link  |  
  15. Azab, M.E., E.M. Flefel, N.M. Sabry and A.E.E. Amr, 2016. Synthesis and antimicrobial activity of some linear dipeptide pyridine and macrocyclic pentaazapyridine candidates. Z. Naturforsch, 71: 803-810.
    CrossRef  |  Direct Link  |  
  16. Azab, M.E., S.A. Rizk and A.E.E. Amr, 2015. Synthesis of some novel heterocyclic and Schiff base derivatives as antimicrobial agents. Molecules, 20: 18201-18218.
    CrossRef  |  Direct Link  |  
  17. Azab, M.E., A.E.E. Amr and M.A. Al-Omar, 2015. Synthesis of chiral macrocyclic candidates: IV. Synthesis and antimicrobial activity of some tricyclooctacosa(triaconta)hexaene bis-Schiff base derivatives. Russ. J. Gen. Chem., 85: 1952-1958.
    CrossRef  |  Direct Link  |  
  18. Azab, M.E. and A.E.E. Amr, 2015. Synthesis of chiral linear and macrocyclic candidates: III. Synthesis and antimicrobial activity of linear tetrapeptide and macrocyclic pentapeptide Schiff Bases. Russ. J. Gen. Chem., 85: 1513-1521.
    CrossRef  |  Direct Link  |  
  19. Salem, M.A.I., M.E. Azab and I.S.A. Mabrouk, 2014. Action of nitrogen and carbon nucleophiles on benzoxazin-4(H)-one derivative as convenient methods for the synthesis of some novel heterocyclic systems. Int. J. Sci. Eng. Res., 5: 1137-1150.
  20. Khamees, H., G.A. Abdel Jaleel, M.E. Azab, G.A.M. Mohamed and T.A. Abd-elaziz et al., 2013. Synthesis, characterization, anticancer, analgesic, and anti-inflammatory activities of hitherto unknown thiazolo[3,2-A] pyridine and thiazolo [3,2-A] 1,8-naphthyridine derivatives. J. Atoms Mol., 3: 478-491.
    Direct Link  |  
  21. El-Hashash, M.A., M.E. Azab and J.M. Morsy, 2013. A novel series of biologically active quinazolinones through ring transformation of 2-(5-Nitrofuran-2-yl)-4H-benzo[d][1,3]oxazin-4-one. Int. J. Sci. Eng. Res., 4: 218-228.
  22. Azab, M.E., M.M. Youssef and E.A. El-Bordany, 2013. Synthesis and antibacterial evaluation of novel heterocyclic compounds containing a sulfonamido moiety. Molecules, 18: 832-844.
    CrossRef  |  Direct Link  |  
  23. Youssef, A., M.E. Azab and M.M. Youssef, 2012. Bromination and diazo-coupling of pyridinethiones; microwave assisted synthesis of isothiazolopyridine, pyridothiazine and pyridothiazepines. Molecules, 17: 6930-6943.
    CrossRef  |  Direct Link  |  
  24. Mahmoud, M.R., F.A. El-Bassiouny, M.E. Azab, M.Y. El-Kady and H.M. Rashed, 2009. Heteroannulation of chromene derivatives. Synthesis of chromeno[4,3-e]indazolne, chromeno[4,3-f]-quinazoline and pyrano[3,2-c]chromene derivatives. J. Chem. Res., 2009: 41-45.
  25. Madkour, H.M.F., M.E. Azab and M.A.E. Ibraheem, 2009. 5,6,7,8-tetrahydrobenzo[b]thieno [2,3-d] pyrimidine-4(3H) one as a synthon of heterocyclic systems. Bulgarian Chem. Commun., 41: 12-18.
  26. Gaenzler, F.C., C.L. Guo, Y.W. Zhang, M.E. Azab, M.A. Salem, D.P. Fan and M.B. Smith, 2009. 2-Dienylphenacyloxazolones and an intramolecular Diels-Alder approach to the A-B-C ring system of phenanthridone alkaloids. Tetrahedron, 65: 8781-8785.
    CrossRef  |  Direct Link  |  
  27. Azab, M.E., E.A. Kassab, M.A. El-Hashash and R.S. Ali, 2009. Synthesis and antibacterial activity of some new 4(3H) quinazolin-4-one derivatives. Phosphorus Sulfur Silicon Relat. Elements, 184: 610-625.
    CrossRef  |  Direct Link  |  
  28. Salem, M.A.I., H.M.F. Madkour, M.I. Marzouk, M.E. Azab and N.F.H. Mahmoud, 2008. Pyrimidinthiones (part I): Utility of 2-thioxopyrimidin-6-(1H) ones as ring transformer in the synthesis of fused bi-and tri-cyclic heterocyclic compounds and their potential biological activities. Phosphorus Sulfur Silicon Relat. Elements, 183: 2596-2614.
    CrossRef  |  Direct Link  |  
  29. Madkour, H.M.F., M.E. Azab, D.A. Mhanna and M.A. El-Hashash, 2008. Behaviour of dynamic 6,8-dibromo-2-methyl-4-(H)-3,1-benzoxazin-4-one towards some nitrogen nucleophiles: Synthesis of new quinazolinones with anticipated biological activity. Org. Chem. Indian J., 4: 142-149.
  30. Azab, M.E., 2008. Utility of the enaminonitrile moiety in the synthesis of some biologically active thienopyrimidine derivatives. Phosphorus Sulfur Silicon Relat. Elements, 183: 1766-1782.
    CrossRef  |  Direct Link  |  
  31. Mahmoud, M.R., E.A. El-Bordany, M.E. Azab and E.A. Soliman, 2007. Synthesis of new thiadiazoles, 1,2,4-Triazolo[3,4-b]-1,3,4-thiadiazoles and 1,2,4-Triazolo[2,3-c]quinazoline derivatives from 3,1-benzoxazin (4H)-one derivative. Phosphorus Sulfur Silicon Relat. Elements, 182: 1275-1289.
    CrossRef  |  Direct Link  |  
  32. Madkour, H.M.F., M.A.I. Salem, M.I. Marzouk, M.E. Azab and N.F.H. Mahmoud, 2007. Utility of cyanothioacetamide in the synthesis of pyrazolo [4,3-c], isoxazolo[4,5-c], thieno [2,3-b] and furo [2,3-c] of thioxopyridine derivatives and their antibacterial activities. Am.-Eurasian J. Scient. Res., 2: 161-169.
    Direct Link  |  
  33. Azab, M.E., E.A. El-Bourdany, S.S. Abdel-Wahab and E.A. Soliman, 2007. Synthesis of novel pyrazole, pyridazine and pyrimidine derivatives containing sulfonamido moiety. Al-Azhar Univ. Bull. Sci., 18: 167-178.
  34. Azab, M.E., H.M.F. Madkour and M.A.E. Ibraheem, 2006. The utility of 2-(5,6,7,8-Tetrahydrobenzo[b] thieno-[2,3-d]pyrimidin-4-yloxy) acethydrazide in heterocyclic synthesis. Phosphoru, Sulfur Silicon Relat. Elements, 181: 1299-1313.
    CrossRef  |  Direct Link  |  
  35. Salem, M.A.I., E.A. Soliman, M.B. Smith, M.R. Mahmoud and M.E. Azab, 2004. Utility of 1-(2,4-dimethoxyphenyl)-3-aryl-prop-2-ene-1-ones as ring transformer in preparing heterocyclic compounds and their potential biological activities. Phosphorus Sulfur Silicon Relat. Elements, 179: 61-76.
    CrossRef  |  Direct Link  |  
  36. Batterjee, S.M., M.I. Marzouk, M.E. Aazab and M.A. El‐Hashash, 2003. The electrochemistry of some ferrocene derivatives: Redox potential and substituent effects. Applied Organometallic Chem., 17: 291-297.
    CrossRef  |  Direct Link  |  
  37. Azab, M.E., G.A.M.E.H. Ali and A.F. Abdel-Wahab, 2003. Studies on thiazolopyridines-A novel synthesis of bisthiazolopyridines as promising antimicrobial agents. Acta Pharm., 53: 213-221.
    PubMed  |  
  38. Azab, M.E., H.M.F. Madkour and M.R. Mahmoud, 2002. Synthesis and nucleophilic reactions of N-(1-naphthyl)-3,4-methylenedioxybenzyl-idinehomophthalisoimidium perchlorate. Synthetic Commun., 32: 393-402.
    CrossRef  |  Direct Link  |  
  39. Elgazwy, A.S.S.H. and M.E. Azab, 2001. Synthesis and biological activity of2-thioxo-[1H]-5-spirocyclohexylimidazo[4,3-b] quinazolone and 8-azaquinazolone derivatives. Phosphorus Sulfur Silicon Relat. Elements, 173: 105-113.
    CrossRef  |  Direct Link  |  
  40. Madkour, H.M.F., M.A.I. Salem, T.M. AbdelRahman and M.E. Azab, 1994. Reactions of 5-(p-anisyl)-2-methyl-7-(p-tolyl)-4H-pyrido-[2,3-d][1,3]-oxazin-4-one. Heterocycles, 38: 57-69.